MTX DRUG - SCI & TECH

News: New highly fluorescent material brings non-enzymatic approach for detection of anticancer drug Methotrexate known for toxicity at high dosage

 

What's in the news?

       Scientists of Institute of Advanced Study in Science and Technology (IASST), an autonomous institute of Department of Science and Technology (DST) have developed a highly fluorescent material that can be used as a visual sensing platform for detecting the anti-cancer drug Methotrexate (MTX).

 

Methotrexate (MTX):

       Methotrexate belongs to a class of drugs known as antimetabolite.

       It is used to treat various medical conditions, primarily cancers, autoimmune diseases, and certain inflammatory conditions.

       The MTX overdose in blood plasma is hazardous if it remains in the system for more than 10 hours, resulting in poisoning effects on the lungs, ulcers of the stomach and heart stroke.

 

New highly fluorescent material for detection of MTX:

       This highly fluorescent material has been developed using phosphorene, cystine and gold (Ph-Cys-Au).

       It has exceptional optical properties and thus can be used as a visual sensing platform for detecting the anti-cancer drug MTX overdose.

 

Significance of the discovery:

       The materials are biocompatible with a good detection limit.

       Traditional procedures for detecting overdosage of MTX are relatively more time consuming and involve complex instrumentation.

       The nanocomposite exhibited in vitro cytotoxicity (quality of a substance to be toxic to cells in an artificial, controlled environment outside of a living organism) towards cancerous cells, but it was non-cytotoxic for non-cancerous cells.